Discovery, SAR, and biological evaluation of a novel series of piperazine-based inhibitors of glycine transporter-1 (GlyT-1)

Christopher Cioffi; Shuang Liu; Mark Wolf; Peter Guzzo; Kashinath Sadalapure; Viswewwaran Parthasarathy; Jun-Ho Maeng; Edmund Carulli; David Loong; Xiao Fang; Priya Gupta; Shailijia Panduga; Karunankaran Kalesh; Lakshman Matta; Sue Choo; Ronald Buckle; Randall Davis; Samuel Sakwa; Min Hu; Dattatraya Dethe; Bruce Sargent; Nicholas Moore; Michele Luche; Yuri Khmelnitsky; Jiffry Ismail; Helen Decornez; Douglas Kitchen; Patrick Love; Megan Watson; Janet Adolphson; Godfrey Padilla; Kathryn Waikins; Susan Tom; Anna Ngo; Mark Chung; Mei Bai; Nidhi Johal; Srividya Swaminathan; Andrew Mhyre

Discovery, SAR, and biological evaluation of a novel series of piperazine-based inhibitors of glycine transporter-1 (GlyT-1)

Christopher Cioffi, Shuang Liu, Mark Wolf, Peter Guzzo, Kashinath Sadalapure, Viswewwaran Parthasarathy, Jun-Ho Maeng, Edmund Carulli, David Loong, Xiao Fang, Priya Gupta, Shailijia Panduga, Karunankaran Kalesh, Lakshman Matta, Sue Choo, Ronald Buckle, Randall Davis, Samuel Sakwa, Min Hu, Dattatraya DetheBruce Sargent, Nicholas Moore, Michele Luche, Yuri Khmelnitsky, Jiffry Ismail, Helen Decornez, Douglas Kitchen, Patrick Love, Megan Watson, Janet Adolphson, Godfrey Padilla, Kathryn Waikins, Susan Tom, Anna Ngo, Mark Chung, Mei Bai, Nidhi Johal, Srividya Swaminathan, Andrew Mhyre

Research output: Contribution to journal › Article › peer-review

Original language	English
Journal	ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY
Volume	249
Publication status	Published - 22 Mar 2015
Externally published	Yes

Cite this

Cioffi, C., Liu, S., Wolf, M., Guzzo, P., Sadalapure, K., Parthasarathy, V., Maeng, J-H., Carulli, E., Loong, D., Fang, X., Gupta, P., Panduga, S., Kalesh, K., Matta, L., Choo, S., Buckle, R., Davis, R., Sakwa, S., Hu, M., ... Mhyre, A. (2015). Discovery, SAR, and biological evaluation of a novel series of piperazine-based inhibitors of glycine transporter-1 (GlyT-1). ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 249.

Cioffi, Christopher ; Liu, Shuang ; Wolf, Mark ; Guzzo, Peter ; Sadalapure, Kashinath ; Parthasarathy, Viswewwaran ; Maeng, Jun-Ho ; Carulli, Edmund ; Loong, David ; Fang, Xiao ; Gupta, Priya ; Panduga, Shailijia ; Kalesh, Karunankaran ; Matta, Lakshman ; Choo, Sue ; Buckle, Ronald ; Davis, Randall ; Sakwa, Samuel ; Hu, Min ; Dethe, Dattatraya ; Sargent, Bruce ; Moore, Nicholas ; Luche, Michele ; Khmelnitsky, Yuri ; Ismail, Jiffry ; Decornez, Helen ; Kitchen, Douglas ; Love, Patrick ; Watson, Megan ; Adolphson, Janet ; Padilla, Godfrey ; Waikins, Kathryn ; Tom, Susan ; Ngo, Anna ; Chung, Mark ; Bai, Mei ; Johal, Nidhi ; Swaminathan, Srividya ; Mhyre, Andrew. / Discovery, SAR, and biological evaluation of a novel series of piperazine-based inhibitors of glycine transporter-1 (GlyT-1). In: ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY. 2015 ; Vol. 249.

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title = "Discovery, SAR, and biological evaluation of a novel series of piperazine-based inhibitors of glycine transporter-1 (GlyT-1)",

author = "Christopher Cioffi and Shuang Liu and Mark Wolf and Peter Guzzo and Kashinath Sadalapure and Viswewwaran Parthasarathy and Jun-Ho Maeng and Edmund Carulli and David Loong and Xiao Fang and Priya Gupta and Shailijia Panduga and Karunankaran Kalesh and Lakshman Matta and Sue Choo and Ronald Buckle and Randall Davis and Samuel Sakwa and Min Hu and Dattatraya Dethe and Bruce Sargent and Nicholas Moore and Michele Luche and Yuri Khmelnitsky and Jiffry Ismail and Helen Decornez and Douglas Kitchen and Patrick Love and Megan Watson and Janet Adolphson and Godfrey Padilla and Kathryn Waikins and Susan Tom and Anna Ngo and Mark Chung and Mei Bai and Nidhi Johal and Srividya Swaminathan and Andrew Mhyre",

year = "2015",

month = mar,

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language = "English",

volume = "249",

journal = "ACS National Meeting Book of Abstracts",

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publisher = "American Chemical Society",

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Cioffi, C, Liu, S, Wolf, M, Guzzo, P, Sadalapure, K, Parthasarathy, V, Maeng, J-H, Carulli, E, Loong, D, Fang, X, Gupta, P, Panduga, S, Kalesh, K, Matta, L, Choo, S, Buckle, R, Davis, R, Sakwa, S, Hu, M, Dethe, D, Sargent, B, Moore, N, Luche, M, Khmelnitsky, Y, Ismail, J, Decornez, H, Kitchen, D, Love, P, Watson, M, Adolphson, J, Padilla, G, Waikins, K, Tom, S, Ngo, A, Chung, M, Bai, M, Johal, N, Swaminathan, S & Mhyre, A 2015, 'Discovery, SAR, and biological evaluation of a novel series of piperazine-based inhibitors of glycine transporter-1 (GlyT-1)', ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, vol. 249.

Discovery, SAR, and biological evaluation of a novel series of piperazine-based inhibitors of glycine transporter-1 (GlyT-1). / Cioffi, Christopher; Liu, Shuang; Wolf, Mark; Guzzo, Peter; Sadalapure, Kashinath; Parthasarathy, Viswewwaran; Maeng, Jun-Ho; Carulli, Edmund; Loong, David; Fang, Xiao; Gupta, Priya; Panduga, Shailijia; Kalesh, Karunankaran; Matta, Lakshman; Choo, Sue; Buckle, Ronald; Davis, Randall; Sakwa, Samuel; Hu, Min; Dethe, Dattatraya; Sargent, Bruce; Moore, Nicholas; Luche, Michele; Khmelnitsky, Yuri; Ismail, Jiffry; Decornez, Helen; Kitchen, Douglas; Love, Patrick; Watson, Megan; Adolphson, Janet; Padilla, Godfrey; Waikins, Kathryn; Tom, Susan; Ngo, Anna; Chung, Mark; Bai, Mei; Johal, Nidhi; Swaminathan, Srividya; Mhyre, Andrew.

In: ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, Vol. 249, 22.03.2015.

Research output: Contribution to journal › Article › peer-review

TY - JOUR

T1 - Discovery, SAR, and biological evaluation of a novel series of piperazine-based inhibitors of glycine transporter-1 (GlyT-1)

AU - Cioffi, Christopher

AU - Liu, Shuang

AU - Wolf, Mark

AU - Guzzo, Peter

AU - Sadalapure, Kashinath

AU - Parthasarathy, Viswewwaran

AU - Maeng, Jun-Ho

AU - Carulli, Edmund

AU - Loong, David

AU - Fang, Xiao

AU - Gupta, Priya

AU - Panduga, Shailijia

AU - Kalesh, Karunankaran

AU - Matta, Lakshman

AU - Choo, Sue

AU - Buckle, Ronald

AU - Davis, Randall

AU - Sakwa, Samuel

AU - Hu, Min

AU - Dethe, Dattatraya

AU - Sargent, Bruce

AU - Moore, Nicholas

AU - Luche, Michele

AU - Khmelnitsky, Yuri

AU - Ismail, Jiffry

AU - Decornez, Helen

AU - Kitchen, Douglas

AU - Love, Patrick

AU - Watson, Megan

AU - Adolphson, Janet

AU - Padilla, Godfrey

AU - Waikins, Kathryn

AU - Tom, Susan

AU - Ngo, Anna

AU - Chung, Mark

AU - Bai, Mei

AU - Johal, Nidhi

AU - Swaminathan, Srividya

AU - Mhyre, Andrew

PY - 2015/3/22

Y1 - 2015/3/22

UR - http://gateway.webofknowledge.com/gateway/Gateway.cgi?GWVersion=2&SrcAuth=ORCID&SrcApp=OrcidOrg&DestLinkType=FullRecord&DestApp=WOS_CPL&KeyUT=WOS:000411186502335&KeyUID=WOS:000411186502335

M3 - Article

VL - 249

JO - ACS National Meeting Book of Abstracts

JF - ACS National Meeting Book of Abstracts

SN - 0065-7727

ER -

Discovery, SAR, and biological evaluation of a novel series of piperazine-based inhibitors of glycine transporter-1 (GlyT-1)

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